Force Field X is a group of open source (GPL v. 3), platform independent (Java Runtime Environment) modules for molecular biophysics. Key methods include:
In collaboration with scientists at Vertex Pharmacueticals, we are using the polarizable AMOEBA force field evaluated using Ewald summation to re-refine protein-drug structures in the context of the original diffraction data (ie. using an X-ray likelihood target) in order to provide the most precise atomic resolution models possible.
The Ewald refinements exhibit:
| Original (1YI4, No Electrostatics) | Ewald Refinement of the Binding Pocket |
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| Model | R | Rfree | Clash Score and Percentile | Poor Rotamer | Ramachandram Favored | MolProbity Score and Percentile | Resolution (A) | Structure |
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| Original Refinements | ||||||||
| PIM-1 Bound to Adenosine | 20.22 | 23.49 | 24.91 / 46th | 7.56% | 93.92% | 2.96 / 33rd | 2.4 | 1YI4 |
| Staphylococcus Aureus Gyrase B with Inhibitor | 23.09 | 32.49 | 33.93 / 20th | 5.45% | 94.78% | 2.93 / 28th | 2.3 | 3G75 |
| Janus Kinase Bound to Inhibitor | 22.07 | 28.60 | 18.87 / 54th | 5.75% | 96.80% | 2.55 / 47th | 2.2 | 3KCK |
| Extracellular Signal-Regulated Kinase (ERK2) with Inhibitor | 20.60 | 24.54 | 11.41 / 94th | 3.65% | 97.26% | 2.14 / 92nd | 2.5 | 3I60 |
| Ewald Refinements | ||||||||
| PIM-1 Bound to Adenosine | 17.76 | 22.37 | 3.42 / 99th | 7.08% | 95.85% | 2.07 / 91rst | 2.4 | 1YI4_Ewald.pdb |
| Staphylococcus Aureus Gyrase B with Inhibitor | 20.64 | 30.48 | 3.74 / 99th | 5.13% | 93.68% | 2.12 / 85th | 2.3 | 3G75_Ewald.pdb |
| Janus Kinase Bound to Inhibitor | 20.83 | 28.13 | 1.67 / 99th | 4.56% | 97.17% | 1.57 / 93rd | 2.2 | 3KCK_Ewald.pdb |
| Extracellular Signal-Regulated Kinase (ERK2) with Inhibitor | 18.55 | 26.66 | 3.41 / 99th | 4.32% | 96.96% | 1.79 / 98th | 2.5 | 3I60_Ewald.pdb |